DEVELOPMENT OF GREEN PROTOCOLS FOR THE SYNTHESIS OF 1H-BENZO[D]IMIDAZOLO ARYL AMIDE DERIVATIVES AND EVALUATION OF THEIR BIOLOGICAL ACTIVITY - TRƯỜNG ĐẠI HỌC HỒNG ĐỨC

Tìm thấy 10,000 tài liệu liên quan tới tiêu đề "Development of Green protocols for the synthesis of 1H-benzo[d]imidazolo aryl amide derivatives and...":

Synthesis and evaluation of antimicrobial, antitubercular and anticancer activities of 2-(1-benzoyl-1H-benzo[d] imidazol-2-ylthio)-N-substituted acetamides

Synthesis and evaluation of antimicrobial, antitubercular and anticancer activities of 2-(1-benzoyl-1H-benzo[d] imidazol-2-ylthio)-N-substituted acetamides

The study describes the synthesis, characterization, in vitro antimicrobial and anticancer evaluation of a series of 2-(1-benzoyl-1H-benzo[d]imidazol-2-ylthio)-N-substituted acetamide derivatives. The synthesized derivatives were also assessed for in vitro antitubercular activity against Mycobacteri[r]

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Influence of new templating agent for the synthesis of coral-like TiO 2 nanoparticles and their photocatalytic activity

INFLUENCE OF NEW TEMPLATING AGENT FOR THE SYNTHESIS OF CORAL-LIKE TIO 2 NANOPARTICLES AND THEIR PHOTOCATALYTIC ACTIVITY

Fig. 2 XRD patterns of calcined TiO 2 samples, DES-1C (a), DES-2C (b), DES-3C (c) and DES-4C (d).
3.1.1 Influence of concentration of acidic DES on the phase structure of TiO 2
It has been observed from XRD analysis that the

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Green synthesis, characterization and antimicrobial evaluation of nano silver on mastitis causing microorganisms

Green synthesis, characterization and antimicrobial evaluation of nano silver on mastitis causing microorganisms

Nanotechnology is now creating a growing sense of excitement in the field of life science. Nano particles can be synthesized by physical and chemical method but green synthesis method is the most emerging approach of preparation due to eco friendly and less time consuming procedure. This study aimed[r]

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Long non-coding RNA MEG3 inhibits NSCLC cells proliferation and induces apoptosis by affecting p53 expression

Long non-coding RNA MEG3 inhibits NSCLC cells proliferation and induces apoptosis by affecting p53 expression

Long non-coding RNAs play an important role in tumorigenesis, hence, identification of cancerassociated lncRNAs and investigation of their biological functions and molecular mechanisms are important for understanding the development and progression of cancer.

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Summary Of Engineering Doctoral Thesis: Synthesis and cytotoxicity of bengamide analogues A and E

Summary Of Engineering Doctoral Thesis: Synthesis and cytotoxicity of bengamide analogues A and E

The objective of the thesis is to build the synthesis process of Analogs of Bengamide A and E, conduct the biological activity of the synthesized Analogs. To find out more about the details of the content, please consult the thesis summary.

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Summary of chemistry doctoral thesis: Synthesis and identification biological activity of some indenoisoquinoline derivatives

Summary of chemistry doctoral thesis: Synthesis and identification biological activity of some indenoisoquinoline derivatives

The task of the thesis: Synthesis of new derivatives of indenoisoquinoline is based on changes in B ring groups by modifying branching atoms of nitrogen atom and binding of triazole-containing hybrid compounds. Synthesis of new derivatives of indenoisoquinoline based on the change of substituents i[r]

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Summary of chemistry doctoral thesis: Synthesis and identification biological activity of some indenoisoquinoline derivatives

Summary of chemistry doctoral thesis: Synthesis and identification biological activity of some indenoisoquinoline derivatives

The task of the thesis: Synthesis of new derivatives of indenoisoquinoline is based on changes in B ring groups by modifying branching atoms of nitrogen atom and binding of triazole-containing hybrid compounds. Synthesis of new derivatives of indenoisoquinoline based on the change of substituents i[r]

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Synthesis, molecular docking and biological evaluation of bis-pyrimidine Schiff base derivatives

Synthesis, molecular docking and biological evaluation of bis-pyrimidine Schiff base derivatives

Heterocyclic pyrimidine nucleus, which is an essential base component of the genetic material of deoxyribonucleic acid, demonstrated various biological activities. A series of bis-pyrimidine Schiff bases were synthesized and screened for its antimicrobial and anticancer potentials.

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Summary of chemistry doctoral thesis: Synthesis and bioactivity evaluation of new vinca alkaloid derivatives

Summary of chemistry doctoral thesis: Synthesis and bioactivity evaluation of new vinca alkaloid derivatives

The objectives of the thesis: Synthesis of new vinca alkaloid derivatives containing different substituents on C-3'' and N-6'' positions in ring D of the velbanamine subunit, concurrently evaluating the biological activity of the derivatives synthesized.

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SYNTHESIS OF GUANIDINO ANALOGUES AS POTENTIAL NITRIC OXIDE SYNTHASE INHIBITORS

SYNTHESIS OF GUANIDINO ANALOGUES AS POTENTIAL NITRIC OXIDE SYNTHASE INHIBITORS


44 of L-Arg is absent in the case of L-NIO, probably due to the increased hydrophobicity upon L-NIO binding.
The binding of L-NPA ( 07 ) 176 , known as nNOS selective, is similar to that of L-Arg. The propyl group is directed towards <[r]

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CẨM NANG BÓNG ĐÁ

104 Synthesis of N1-Benzyl-N2-nitroguanidines Biological Evaluation of N1-Benzyl-N2-nitroguanidines CHAPTER 10 FURTHER INVESTIGATIONS USING GUANIDINO-CONTAINING COMPOUNDS 112 Synthesis a[r]

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The relationship between motor proficiency and reading ability in Year 1 children: A cross-sectional study

The relationship between motor proficiency and reading ability in Year 1 children: A cross-sectional study

Movement and physical activity is crucial to brain development and has a positive impact on the ability to learn. With children spending a large portion of their time in the school setting, physical activity and the development of motor skills in this environment may not only impact their overall de[r]

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Design and synthesis of novel 3-(thiophen-2-yl)-1,5-dihydro-2H-pyrrol-2-one derivatives bearing a hydrazone moiety as potential fungicides

Design and synthesis of novel 3-(thiophen-2-yl)-1,5-dihydro-2H-pyrrol-2-one derivatives bearing a hydrazone moiety as potential fungicides

Tetramic acid, thiophene and hydrazone derivatives were found to exhibit favorable antifungal activity. Aiming to discover novel template molecules with potent antifungal activity, a series of novel 3-(thiophen-2-yl)-1,5-dihydro-2H-pyrrol-2-one derivatives containing a hydrazone group were designed,[r]

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Synthesis, characterization, X-ray structure, computational studies, and bioassay of novel compounds combining thiophene and benzimidazole or 1,2,4-triazole moieties

Synthesis, characterization, X-ray structure, computational studies, and bioassay of novel compounds combining thiophene and benzimidazole or 1,2,4-triazole moieties

Due to their interesting and versatile biological activity, thiophene-containing compounds have attracted the attention of both chemists and medicinal chemists. Some of these compounds have anticancer, anti‑ bacterial, antiviral, and antioxidant activity.

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Evaluation and efficacy of the antibacterial activity of silver and gold nanoparticles synthesize from Camelus dromedarius (Camel) milk against oral pathogenic bacteria

Evaluation and efficacy of the antibacterial activity of silver and gold nanoparticles synthesize from Camelus dromedarius (Camel) milk against oral pathogenic bacteria

The unique property of the silver and gold nanoparticles having antibacterial activity drags the major attention towards the present nanotechnology. Synthesis of nanobodies is of great interest in the development of nanotechnological tool for biomedical applications. This study investigates a compet[r]

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GREEN SYNTHESIS OF METALLIC NANOPARTICLES USING AQUEOUS PLANT EXTRACT AND THEIR ANTIBACTERIAL ACTIVITY

GREEN SYNTHESIS OF METALLIC NANOPARTICLES USING AQUEOUS PLANT EXTRACT AND THEIR ANTIBACTERIAL ACTIVITY

The bio molecules present in plants can act as capping and reducing agents and thus increase the rate of reduction and stabilization of nanoparticles. Biosynthesized metal nanoparticles are more stable in nature and their rate of synthesis is faster than other methods. The present study describes th[r]

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Synthesis, structural determination and antimicrobial evaluation of two novel CoII and ZnII halogenometallates as efficient catalysts for the acetalization reaction of aldehydes

Synthesis, structural determination and antimicrobial evaluation of two novel CoII and ZnII halogenometallates as efficient catalysts for the acetalization reaction of aldehydes

Complexes of imidazole derivatives with transition metal ions have attracted much attention because of their biological and pharmacological activities, such as antimicrobial, antifungal, antiallergic, antitumoural and antimetastatic properties.

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Synthesis and biological activity of myricetin derivatives containing 1,3,4-thiadiazole scafold

Synthesis and biological activity of myricetin derivatives containing 1,3,4-thiadiazole scafold

Myricetin and 1,3,4-thiadiazole derivatives were reported to exhibit favorable antiviral and antibacterial activities. Aiming to discover novel myricetin analogues with potent activities, a series of novel myricetin derivatives containing 1,3,4-thiadiazole moiety were synthesized, and their antibact[r]

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Synthesis and Evaluation of Pyrazine Derivatives with Herbicidal Activity

SYNTHESIS AND EVALUATION OF PYRAZINE DERIVATIVES WITH HERBICIDAL ACTIVITY

Novel pyrazine-sulfonylcarbamates and thiocarbamates (Fig. 3, XIII) (where Z is oxygen or sulfur and R is C1-C4 alkyl, phenyl or benzyl; whereas the pyrazine ring may be variously further substituted) have been found to be good selective herbicides and therefore they ar[r]

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Eugenol derivatives: Synthesis, characterization, and evaluation of antibacterial and antioxidant activities

Eugenol derivatives: Synthesis, characterization, and evaluation of antibacterial and antioxidant activities

Eugenol is the major component of clove essential oil and has demonstrated relevant biological potential with wellknown antimicrobial and antioxidant action. Therefore, this work carried out the synthesis, purification, characterization, and evaluation of the antioxidant and antibacterial potential[r]

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